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CYP2J2 (h), CYP2J2 (h)

Cat#: 400-0879
Species: Human
RegionHuman recombinant
Substratebenzyloxymethyloxy-4-trifluorocoumarin
Substrate [M]10E-6
Km (enzyme affinity)12E-6 M
Vmax0.44 pmol product/pmol CYP2J2(h) /min
ReactionBOMFC + NADPH > 7HFC + NADP
MethodFluorescence
Reference CompoundKetoconazole
IC50 = 140 nM
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