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Kinase, Lipid, PI3Ka (p110a/p85a) (h)

Cat#: 200-0924
Species: Human
RegionHuman recombinant
Enzyme FamilyLipid Kinase
SubstrateFluorescein-labeled PIP2 (phosphoinositol (4,5)bisphosphate)
Substrate [M]2.0E-6M
Km (enzyme affinity)3.8E-6M
Km (ATP)73E-6M
ATP [M]73E-6M
ReactionFluorescein-PIP2 + ATP -> fluorescein-PIP3 + ADP
MethodFluorescence – electrophoretic mobility shift
MeasurementSeparation of phosphorylated and unphosphorylated substrate
Reference CompoundPI-103
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