Retinoic Acid, RARa, Antagonist (h)
| Cat#: | 100-0907 |
| Species: | Human |
| Region | Human recombinant RAR Ligand Binding Domain GST tagged |
| Substrate | 4-[E-2-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl]benzoic acid (TTNPB) |
| Kd (binding affinity) | 2 nM |
| Reaction | Ligand dependent binding of receptor to cofactor |
| Method | Time-Resolved Fluorescence Resonance Energy Transfer |
| Reference Compound | BMS 453 |
